Cenicriviroc

• CAS: 497223-25-3
• Catalog Number: ACM497223253
• Category: Inhibitors
• Molecular Weight: 0
• Description: Cenicriviroc (TAK-652) is an orally active, dual CCR2/CCR5 antagonist, also inhibits both HIV-1 and HIV-2, and displays potent anti-inflammatory and antiinfective activity.
• Synonyms: Cenicriviroc;TAK652

Custom Q&A

What is the molecular formula of cenicriviroc?

The molecular formula of cenicriviroc is C41H52N4O4S.

What is the molecular weight of cenicriviroc?

The molecular weight of cenicriviroc is 696.9 g/mol.

What are some synonyms for cenicriviroc?

Some synonyms for cenicriviroc include TBR-652, TAK-652, and TBR652.

What is the role of cenicriviroc as described in the reference?

Cenicriviroc is described as a chemokine receptor 5 antagonist, an anti-HIV agent, a chemokine receptor 2 antagonist, an antirheumatic drug, and an anti-inflammatory agent.

What class of benzazocines does cenicriviroc belong to?

Cenicriviroc belongs to the class of benzazocines.

What is the IUPAC name of cenicriviroc?

The IUPAC name of cenicriviroc is (5E)-8-[4-(2-butoxyethoxy)phenyl]-1-(2-methylpropyl)-N-[4-[(S)-(3-propylimidazol-4-yl)methylsulfinyl]phenyl]-3,4-dihydro-2H-1-benzazocine-5-carboxamide.

How does cenicriviroc work as an immunomodulating agent?

Cenicriviroc is a dual inhibitor of human C-C chemokine receptor types 2 and 5, which inhibits the activation of CCR2/CCR5-mediated signal transduction pathways, leading to the inhibition of inflammatory processes.

What is the InChIKey of cenicriviroc?

The InChIKey of cenicriviroc is PNDKCRDVVKJPKG-WHERJAGFSA-N.

What is another identifier for cenicriviroc besides CAS and UNII numbers?

Cenicriviroc is also identified by the ChEMBL ID (CHEMBL2110727).

In what trials has cenicriviroc been studied?

Cenicriviroc has been studied in trials focusing on the treatment of HIV-infection/AIDS, AIDS Dementia Complex, Nonalcoholic Steatohepatitis, Human Immunodeficiency Virus, and HIV-1-Associated Cognitive Motor Complex.