1-(4-Pyridinmethyl)pyrazole-4-boronic acid pinacol ester

• CAS: 864754-20-1
• Catalog Number: ACM864754201-1
• Category: Other

Synthetic Use

Upstream Synthesis Route 1

• 10445-91-7
• 269410-08-4

• 864754-20-1

Reference: [1]Current Patent Assignee: ASTRAZENECA PLC - WO2006/20879, 2006, A1
Location in patent: Page/Page column 109
[2]Charoensutthivarakul, Sitthivut; Thomas, Sherine E.; Curran, Amy; Brown, Karen P.; Belardinelli, Juan M.; Whitehouse, Andrew J.; Acebrón-García-de-Eulate, Marta; Sangan, Jaspar; Gramani, Subramanian G.; Jackson, Mary; Mendes, Vitor; Floto, R. Andres; Blundell, Tom L.; Coyne, Anthony G.; Abell, Chris
[ACS Infectious Diseases, 2022, vol. 8, # 2, p. 296 - 309]

Downstream Synthesis Route 1

• 864754-20-1
• 1334167-41-7

• 1334166-50-5

Reference: [1]Bartolomé-Nebreda, José Manuel; Delgado, Francisca; Martín-Martín, María Luz; Martínez-Viturro, Carlos M.; Pastor, Joaquín; Tong, Han Min; Iturrino, Laura; Macdonald, Gregor J.; Sanderson, Wendy; Megens, Anton; Langlois, Xavier; Somers, Marijke; Vanhoof, Greet; Conde-Ceide, Susana
[Journal of Medicinal Chemistry, 2014, vol. 57, # 10, p. 4196 - 4212]

* For details of the synthesis route, please refer to the original source to ensure accuracy.